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Modern Technologies for Synthesizing Drug Substances: Toward Highly Efficient Drug Production
Narkevich I.A., Tarasov I.N., Golant Z.M., Alekhin A.V.
Syntheses of Melanotan II and YSL Amide by Ajiphase® Methodology
Sanguliya T.A., Antipova A.O., Shkavrov S.V., Épshtein N.B.
An Effective and Convenient Process for the Preparation of Ticagrelor: Optimized by Response Surface Methodology and One-Pot Reaction
Wang L., Liu J.
Microwave-Assisted Synthesis, In Vivo Anti-Inflammatory and In Vitro Anti-Oxidant Activities, and Molecular Docking Study of New Substituted Schiff Base Derivatives
Hanif M., Hassan M., Rafiq M., Abbas Q., Ishaq A., Shahzadi S., Seo S., Saleem M.
Stereoselective Transformation of Chiral Amine: Novel Approach to the Synthesis of Optically Active Intermediate of Silodosin
Buchi Reddy R., More K.R., Gupta L.
Synthesis and Pharmacological Potential of New 3-Mercapto-4-Amino(Pyrrolyl-1)-5-(Thienyl-2)-1,2,4-Triazole(4H) Derivatives
Saidov N.B., Georgiyants V.A., Lipakova E.Y.
Using Bioisosteric Replacements to Enhance the Analgesic Properties of 4-Hydroxy-6,7-Dimethoxy-2-oxo-1,2-Dihydroquinoline-3-Carboxamides
Ukrainets I.V., Mospanova E.V., Davidenko A.A.
Synthesis and Antibacterial Activity of 3,6-Diaryl-7H-[1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazines
Iradyan M.A., Iradyan N.S., Minasyan N.S., Paronikyan R.V., Stepanyan G.M.
Synthesis and Pharmacological Activity of 2,9-Disubstituted Imidazo[1,2-a]Benzimidazole Phenyl- and Alkylthiocarbamides
Anisimova V.A., Zhukovskaya O.N., Spasov A.A., Kuznetsova V.A., Kosolapov V.A., Yakovlev D.S., Solov’eva O.A., Sorotskii D.V., Brigadirova A.A., Vorob’ev E.S.
Development of Drug Substances of the Original Class III Antiarrhythmic Drugs Nibentan and Niferidyl
Davydova N.K.
Synthesis, Affinity for Central Benzodiazepine Receptors, and Hypnosedative and Anxiolytic Properties of 3-Acyloxy-5-Aryl-7-Bromo-1,2-Dihydro-3H-1,4-Benzodiazepin-2-Ones
Pavlovsky V.I., Karaseva T.L., Semenishina E.A., Andronati K.S., Yurpalova T.A., Onufrienko O.V., Krivenko Y.R., Krys’ko A.A., Andronati S.A.
Efficient Synthesis of 21-Acetoxypregna-1,4,9(11),16-Tetraene-3,20-Dione, a Key Intermediate in the Synthesis of Highly Active Fluorinated Corticosteroids from 9α-Hydroxyandrostenedione
Andryushina V.A., Stytsenko T.S., Karpova N.V., Yaderets V.V., Dzhavakhiya V.V.
Acetoxybenzoylglycylglycines as Potential Cerebroprotective Compounds
Brel’ A.K., Tyurenkov I.N., Lisina S.V., Popov S.S., Verkholyak D.V., Budaeva Y.N., Volotova E.V., Atapina N.V., Kurkin D.V.
Kilogram-Scale Pilot Synthesis of Fingolimod
Balaev A.N., Busel A.A., Fedorov V.E.
Studying Newly Synthesized and Developed 4-Hydroxy-3-Methoxybenzaldehyde Schiff Bases by UV Spectrophotometry and High Performance Liquid Chromatography
Chigurupati S., Muralidharan S., Cin L.S., Raser W.Y., Santhi K., Kesavanarayanan K.S.
Synthesis and Immunotropic Activity of Quinazolin-4(3H)-One Carbonyl Derivatives
Samotrueva M.A., Tsibizova A.A., Ozerov A.A., Luzhnova S.A., Glukhova E.G., Tyurenkov I.N.
Synthesis and Neurotropic Activity of New Pyrano[3,4-b]Furo[2,3-b]Pyridine Derivatives
Dabaeva V.V., Bagdasaryan M.R., Noravyan A.S., Kazaryan Z.V., Dzhagatspanyan I.A., Nazaryan I.M., Akopyan A.G.
Synthesis, Properties, Analgesic and Anti-Inflammatory Activity, And Hemostatic Effect of 4-Acyl-1-(2-Aminopropyl)- 5-Aryl-3-Hydroxy-3-Pyrrolin-2-Ones and their Derivatives
Gein V.L., Kasimova N.N., Chashchina S.V., Starkova A.V., Syropyatov B.Y.
Synthesis and Pharmacological Activity of C(2)-Substituted Benzimidazoles
Zhukovskaya O.N., Spasov A.A., Yakovlev D.S., Kosolapov V.A., Mal’tsev D.V., Morkovnik A.S., Babkova V.A., Brigadirova A.A., Agatsarskaya Y.V., Taran A.S., Miroshnikov M.V., Sultanova K.T., Kornilov V.I., Anisimova V.A.
Optimization of the First Step of Enoxaparin Synthesis by Hydrolytic Depolymerization of Unfractionated Heparin
Frumin L.E., Yur’eva K.P., Askretkov A.D., Prokhorov D.I., Matveev A.V., Zhavoronok E.S., Panov A.V., Shatalov D.O., Shnyak E.A., Kedik S.A.
Solvent-Free Synthesis and Antibacterial Evaluation of Novel Coumarin Sulfonamides
Mostajeran N., Arshad F.A., Aliyan H., Massah A.R.
N-Substituted 1H-Pyrimidin-4-One Derivatives Possessing Anxiolytic Activity
Oganesyan É.T., Kodonidi I.P., Bandura A.F., Sochnev V.S., Manvelyan É.A., Sysa V.Y.
New Synthesis and Analgesic and Diuretic Activity of Halo-Substituted 4-Hydroxy-1-Methyl-2,2-Dioxo- 1H-2λ6,1-Benzothiazine-3-Carboxanilides
Ukrainets I.V., Petrushova L.A., Dzyubenko S.P., Grinevich L.A.
Synthesis and Neurotropic Activity of Amino Derivatives of Cyclopenta[4′,5′]pyrido[3′,2′:4,5]thieno[3,2-d ]pyrimidines and Pyrimido[4′,5′:4,5]thieno[2,3-c]isoquinolines
Paronikyan E.G., Dashyan S.S., Noravyan A.S., Dzhagatspanyan I.A., Paronikyan R.G., Nazaryan I.M., Akopyan A.G.
Synthesis and Antibacterial Activity of Bis-[1-(Adamantan-1-Yl)Ethyl]Amine Hydrochloride
Krylov V.I., Moiseev S.V., Kutin A.A., Sakhno N.G., Gunar O.V., Yashkir V.A., Merkulov V.A.
Synthesis and Antiglycation Activity of Novel S-Carboxyalkyl Derivatives of 2-Thiouracil
Spasov A.A., Geisman A.N., Kosolapov V.A., Babkov D.A., Rashchenko A.I., Babkova V.A., Zakhar’yashcheva O.Y., Ozerov A.A.
Synthesis and Antimicrobial Activity of 3-Phenyl-1-Methylquinolin-2-One Derivatives
Elenich O.V., Lytvyn R.Z., Blinder O.V., Skripskaya O.V., Lyavinets O.S., Pitkovych K.E., Obushak M.D., Yagodinets P.I.
Synthesis and Antimicrobial, Antiprotozoal, and Fungistatic Activity of [5-(Amino-, Acylamino-, and 2-Pyridylmethylamino)-1-Alkylbenzimidazol-2-yl]Diphenylmethanols
Koshchienko Y.V., Drobin Y.D., Zubenko A.A., Timoshevskii D.A., Fetisov L.N., Bodryakov A.N.
Synthesis and Antidepressant Properties of 3-Methyl-7-(1,1-Dioxothietan-3-YL)-8-Cyclohexylamino-1-Ethyl-1H-Purine-2,6(3H,7H)-Dione
Khaliullin F.A., Shabalina Y.V., Davlyatova G.G., Valeeva L.A.
Analysis of Problems Hindering Implementation of Modern Drug Technologies: Searching for Possible Solutions
Narkevich I.A., Golant Z.M., Semin A.A., Kartashova N.S., Teslev A.A.
Synthesis and Antimicrobial Activity of Thiocyanatoarylation Products of Acrylamide and Methacrylamide by Diphenyl- and Phenylene-Bis-Diazonium Salts
Grishchuk B.D., Yatsyuk V.N., Baranovskii V.S., Pokryshko E.V., Klimnyuk S.I.
Synthesis and Cytotoxic Activity of (4-Substituted-benzylidene)-(3-Phenyl-1,2,4-Oxadiazol-5-YL)Methylamines
Kucukoglu K., Tugrak M., Demirtas A., Sakagami H., Gul H.I.
Synthesis and Antimycobacterial Activity of 5-(Arylmethylene)Hexahydropyrimidine-2,4,6-Triones
Luzhnova S.A., Tyrkov A.G., Gabitova N.M., Yurtaeva E.A.
Synthesis and Anticholinesterase Activity Evaluation of Asymmetric Azines
Figueredo A.S., Queiroz J.E., Dias L.D., Vidal H.D., Machado I.V., Vila Verde G.M., Aquino G.L.
R-Benzylidenehydrazides of NH-Furoyl-5-Iodoanthranilic Acids: Synthesis, Properties, and Analgesic and Antibacterial Activity
Gazizova A.F., Kurbatov E.R., Makhmudov R.R., Bobyleva A.A., Korkodinova L.M., Kurbatova A.A.
Synthesis and some Pharmacological Properties of an Immunoactive Lysine-Containing Tetrapeptide
Kholnazarov B.M., Bobizoda G.M., Olefir Y.V., Prokof’ev A.B., Sapovskii M.M., Evteev V.A., Bunyatyan N.D.
Synthesis, Characterization, Pharmacokinetics and Evaluation of Cytotoxicity for Docetaxel-Oleate Conjugate Targeting MCF-7 Breast Cancer Cells
Bhatia N.M., Kulkarni P.K., Ashtekar S.S., Mahuli D.V., Bhatia M.S.
Synthesis of New 7-bromo-5-(2’-chlorophenyl)-3-arylamino-1,2-dihydro-3H-1,4-benzodiazepine Derivatives and Their Influence on Appetite in Rats
Karaseva T.L., Likhota E.B., Krivenko Y.R., Semibrat’ev S.A., Pavlovskii V.I.
Synthesis and Fungi/Bactericidal Activities of 4-(4-Dimethylaminophenyl)Pyridine Derivatives
Lomov D.A., Abramyants M.G., Astashkina N.V., Korotkikh N.I., Lubenets V.I., Novikov V.P., Komarovskaya-Porokhnyavets E.Z., Smolyar N.N.
Synthesis, Structure, and Analgesic Properties of Phosphorylated Dihydro-1,4-Benzodiazepin-2-Ones*
Pavlovskii V.I., Gololobov Y.G., Andronati S.A., Voronenko E.V., Kabanova T.A., Khalimova E.I., Krasnova I.Y., Khrustalev V.N.
Synthesis and Cytotoxic Activity of Hydroxy-Substituted Glaucocalyxin A
Xiang Z., Wu X., Zheng X.
Kinetics of One-Step Mepivacaine Synthesis on Polymers Containing Pd-Nanoparticles
Abdullaev M.G.
Synthesis, Structure, and Analgesic Activity of Picolylamides of 2-Hydroxy-4-Oxo-4H-Pyrido-[1,2-a]Pyrimidine-3-Carboxylic Acids
Ukrainets I.V., Bereznyakova N.L., Sim G., Davidenko A.A.
Synthesis and Biological Activity of β-Aroylacrylate Salts
Khachikyan R.D., Ovakimyan Z.G., Mikaelyan A.A., Paronikyan R.V., Stepanyan G.M.
Synthesis and Analgesic and Antibacterial Activity of 5-aryl-4-aroyl-1-(4-acetylaminosulfonylphenyl)-3-hydroxy-3-pyrrolin-2-ones
Gein V.L., Bobrovskaya O.V., Seliverstov G.V., Makhmudov R.R., Novikova V.V.
Synthesis, Antimicrobial and In Silico EGFR Inhibitory Activity Evaluation of Sulfonylamino Pyrrolidine Derivatives
Kumar B.S., Prasad A.R., Reddy P.R., Ravindranath L.K.
Convenient Four-Step Synthesis of H-Pyr-His-Trp-OH, a Key Tripeptide Intermediate for the Production of Synthetic Gonadoliberin Agonists
Balaev A.N., Okhmanovich K.A., Fedorov V.E.
1-Substituted 2-Benzylaminobenzimidazoles with Phenyl Methoxyls: Synthesis, Computer Prediction, and Pharmacological Activity
Zhukovskaya O.N., Anisimova V.A., Spasov A.A., Vasil’ev P.M., Kosolapov V.A., Kucheryavenko A.F., Gurova N.A., Naumenko L.V., Kuznetsova V.A., Sorotskii D.V., Solov’eva O.A., Reznikov E.V., Gurova V.V., Sirotenko V.S.
N-(5-(Trifluoromethyl)-1,3,4-Thiadiazol-2-Yl)Benzamide and Benzothioamide Derivatives Induce Apoptosis Via Caspase-Dependent Pathway
Aliabadi A., Afnanzade N., Hosseinzadeh L., Mohammadi-Farani A., Shafiee M.H., Nazari H., Ahmadi F., Foroumadi A.
Synthesis and Neurotropic Activity of New Condensed Pyrano[4,3-b]-Pyridines Derivatives
Dabaeva V.V., Bagdasaryan M.R., Dashyan S.S., Dzhagatspanyan I.A., Nazaryan I.M., Akopyan A.G., Paronikyan R.G.
Reductive Amination of Sterically Hindered Arylaminoketones Using a Modified Leuckart Reaction
Skachilova S.Y., Zheltukhin N.K., Sergeev V.N., Davydova N.K.
Facile One-Pot Synthesis Methodology for Nitrogen-Containing Heterocyclic Derivatives of 3,5-Disubstituted 4,5-Dihydro-1H-Pyrazole, Their Biological Evaluation and Molecular Docking Studies
Upadhyay S., Tripathi A.C., Paliwal S., Saraf S.K.
The Search for Pharmacologically Active Compounds Among the 2-Dialkylaminobenzimidazoles
Zhukovskaya O.N., Anisimova V.A., Spasov A.A., Yakovlev D.S., Gurova N.A., Kucheryavenko A.F., Salaznikova O.A., Kuznetsova V.A., Mal’tsev D.V., Brigadirova A.A., Morkovina Y.V., Solov’eva O.A., Gurova V.V., Reznikov E.V.
Synthesis and Antimicrobial Activity of 5-(Heterylmethylene)Hexahydropyrimidin-2,4,6-Triones
Tyrkov A.G., Sukhenko L.T., Yurtaeva E.A.
Synthesis and Antiviral Activity of Hydroxy-Substituted Benzaldehydes and Related Compounds
Shadyro O.I., Sorokin V.L., Ksendzova G.A., Savinova O.V., Samovich S.N., Pavlova N.I., Polozov G.I., Boreko E.I.
Design, Synthesis and Cytotoxicity Evaluation of N-(5-Benzylthio)-4H-1,2,4-Triazol-3-YL)-4-Fluorobenzamide Derivatives as Potential Anticancer Agents
Aliabadi A., Mohammadi-Frarni A., Azizi M., Ahmadi F.
Cytotoxicity of New Ferulic-Acid Derivatives on Human Colon Carcinoma (HCT116) Cells
Bakholdina L.A., Markova A.A., Khlebnikov A.I., Sevodin V.P.
Modification of the Benzene Moiety in the Quinolone Nucleus of 4-Hydroxy-6,7-Dimethoxy-2-Oxo-N-(Pyridin-3-Ylmethyl)-1,2-Dihydroquinoline-3-Carboxamide as an Attempt to Enhance its Analgesic Activity
Ukrainets I.V., Mospanova E.V., Bereznyakova N.L., Davidenko A.A.
Synthesis and Antimicrobial Activity of 5-(Arylmethylidene)-2,4,6-Pyrimidine-2,4,6(1H,3H,5H)-Triones
Luzhnova S.A., Tyrkov A.G., Gabitova N.M., Yurtaeva E.A.
Synthesis and Biological Properties of {[(4-Hydroxy-1-Methyl-2,2-Dioxido-1H-2,1-Benzothiazin-3-YL)Carbonyl]Amino}-Benzoic Acids and Their Derivatives
Ukrainets I.V., Petrushova L.A., Dzyubenko S.P., Grinevich L.A., Sim G.
Synthesis of Carbazole Derivative PLX01107 and its Pharmacokinetics for Various Administration Routes in CD-1 Mice
Eremina N.V., Kazei V.I., Purmal A.A., Durnev A.D.
Synthesis, Structural Characterization and Cancer Cell Cytotoxic Activity of Vadimezan Hydrazones
Zhang S., Xu F., Ge Q., Li H., Hu W.
Synthesis and Antibacterial Activity of 3,4-Diaryl-5-(4-Guanidylsulfonylphenyl)-4,6-Dihydropyrrolo[3, 4-C]Pyrazol-6-Ones
Bobrovskaya O.V., Kovtonogova I.V., Gein V.L., Gein L.F., Odegova T.F.
Synthesis and Antibacterial and Immunobiological Activity of Ethyl-1-(4-Aminosulfonylphenyl)-5-Aryl-3-Hydroxy-2-Oxo-3-Pyrroline-4-Carboxylates
Gein V.L., Bobrovskaya O.V., Odegova T.F., Krylova I.V., Gein O.N., Sopova E.É., Gein S.V.
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