Issue |
Title |
File |
Vol 53, No 9 (2019) |
Synthesis and Cardiotropic Activity of 1-(Methoxybenzyl)-4-{2-[(Methoxybenzyl)-Amino]Ethyl}Piperazines |
(Eng)
|
Mokrov G.V., Likhosherstov A.M., Barchukov V.V., Stolyaruk V.N., Tsorin I.B., Vititnova M.B., Rebeko A.G., Kryzhanovskii S.A., Gudasheva T.A.
|
Vol 53, No 8 (2019) |
Synthesis and Antitumor and Antimetastatic Activity of 5-hydroxypyrimidine Derivatives |
(Eng)
|
Nikitin S.V., Kovalenko L.P., Rebeko A.G., Zhurikov R.V., Ivanova E.A., Durnev A.D.
|
Vol 53, No 7 (2019) |
Synthesis and Cardiotropic Activity of Cyclic Methoxyphenyltriazaalkanes |
(Eng)
|
Mokrov G.V., Likhosherstov A.M., Barchukov V.V., Stolyaruk V.N., Tsorin I.B., Vititnova M.B., Rebeko A.G., Kryzhanovskii S.A., Gudasheva T.A.
|
Vol 53, No 6 (2019) |
Synthesis and In Vitro Neuroprotective Activity of Analogs with Various Spacer Lengths of a Dimeric Dipeptide Mimetic (GK-2) of Nerve Growth Factor |
(Eng)
|
Tarasyuk A.V., Sazonova N.M., Kurilov D.V., Lubin A.A., Antipova T.A., Gudasheva T.A.
|
Vol 53, No 5 (2019) |
Synthesis and In Vivo Evaluation of New Coumarin Conjugates as Potential Indirect-Action Anticoagulants |
(Eng)
|
Bang N.C., Abyshev A.Z., Ivkin D.Y.
|
Vol 53, No 4 (2019) |
Water-Soluble Anionic C60-Fullerene Derivatives as Antidotes for HG(II) Ions in Tests on Escherichia Coli Cells |
(Eng)
|
Zhilenkov A.V., Khakina E.A., Troshin P.A., Karimov I.F., Deryabin D.G.
|
Vol 53, No 3 (2019) |
Synthesis and Anticonvulsant Activity of 4-Amino-3-Nitro-1-Thiocoumarins and 4-Amino-3-Nitroquinolin-2-Ones |
(Eng)
|
Mokrov G.V., Voronina T.A., Litvinova S.A., Kovalev I.G., Nerobkova L.N., Durnev A.D., Gudasheva T.A., Seredenin S.B.
|
Vol 53, No 2 (2019) |
Synthesis of C5-C6 Derivatives of 1,3-Dimethyl-5-Fluorouracil and 5-Fluorouracil. Screening for Antiviral Activity |
(Eng)
|
Chernikova I.B., Khursan S.L., Eropkin M.Y., Yunusov M.S.
|
Vol 53, No 1 (2019) |
Design and Antitumor Activity of Platinum Complexes |
(Eng)
|
Kritchenkov A.S., Stanishevskii Y.M., Skorik Y.A.
|
Vol 52, No 12 (2019) |
R-Benzylidenehydrazides of NH-Furoyl-5-Iodoanthranilic Acids: Synthesis, Properties, and Analgesic and Antibacterial Activity |
(Eng)
|
Gazizova A.F., Kurbatov E.R., Makhmudov R.R., Bobyleva A.A., Korkodinova L.M., Kurbatova A.A.
|
Vol 52, No 11 (2019) |
Polyene Macrolide Antibotic Derivatives: Preparation, Overcoming Drug Resistance, and Prospects for Use in Medical Practice (Review) |
(Eng)
|
Belakhov V.V., Garabadzhiu A.V., Chistyakova T.B.
|
Vol 52, No 10 (2019) |
Synthesis and Antiviral Activity of Polycyclic N-Amidoimides Based on 4-Oxatetracyclo-[5.3.2.02, 6.08, 10]Dodec-11-Ene-3,5-Dione |
(Eng)
|
Selivanov B.A., Bormotov N.I., Shishkina L.N., Belanov E.F., Serova O.A., Kabanov A.S., Mazurkov O.Y., Tikhonov A.Y.
|
Vol 52, No 9 (2018) |
Computer Prediction of Adverse Drug Effects on the Cardiovascular System |
(Eng)
|
Ivanov S.M., Lagunin A.A., Filimonov D.A., Poroikov V.V.
|
Vol 52, No 8 (2018) |
Synthesis and In Vitro Neuroprotector Activity of Diastereoisomers of a Dimeric Dipeptide Mimetic of Nerve Growth Factor GK-2 |
(Eng)
|
Sazonova N.M., Tarasyuk A.V., Shumskii A.N., Rebeko A.G., Antipov P.I., Logvinov I.O., Antipova T.A., Gudasheva T.A.
|
Vol 52, No 6 (2018) |
Structure–Activity (Antihypoxic) Relationship in a Series of Substituted Glyprolines |
(Eng)
|
Kolyasnikova K.N., Kuznetsova E.A., Nikolaev S.V., Antipova T.A., Gudasheva T.A., Seredenin S.B.
|
Vol 52, No 5 (2018) |
Synthesis and Pharmacological Activity of Trifluoromethyl-Containing Imidazo[1,2-A]Benzimidazoles |
(Eng)
|
Zhukovskaya O.N., Spasov A.A., Kuz’menko T.A., Morkovnik A.S., Kucheryavenko A.F., Anisimova V.A., Salaznikova O.A., Gaidukova K.A., Kuznetsova V.A., Babkov D.A., Grechko O.Y., Eliseeva N.V., Rashchenko A.I.
|
Vol 52, No 4 (2018) |
Synthesis and Infarction-Limiting Properties of Peptide Agonists of Opioid Receptors |
(Eng)
|
Tsibul’nikov S.Y., Mukhomedzyanov A.V., Maslov L.N., Ovchinnikov M.V., Sidorova M.V., Kudryavtseva E.V., Bushov Y.V., Lishmanov Y.B., Khaliulin I.
|
Vol 52, No 3 (2018) |
Synthesis and Biological Activity of 2-amino-1-aryl-5-(3,3-dimethyl-2-oxobutylidene)-4-oxo-N-(thiazol-5-yl)-4,5-dihydro-1h-pyrrole-3-carboxamides |
(Eng)
|
Zykova S.S., Igidov N.M., Zakhmatov A.V., Kiselev M.A., Galembikova A.R., Khusnutdinov R.R., Dunaev P.D., Boichuk S.V., Chernov I.N., Rodin I.A.
|
Vol 52, No 2 (2018) |
Synthesis and Cerebrovascular Anti-Ischemic Activity of New 5-Hydroxyadamantan-2-One Derivatives |
(Eng)
|
Kurza E.V., Avdyunina N.I., Gan’shina T.S., Maslennikov D.V., Turilova A.I., Pyatin B.M., Grushevskaya L.N., Zaitseva N.M., Bol’shakova R.F., Kovalev G.I., Vasil’eva E.V., Mirzoyan R.S.
|
Vol 52, No 1 (2018) |
Solvent-Free Synthesis and Antibacterial Evaluation of Novel Coumarin Sulfonamides |
(Eng)
|
Mostajeran N., Arshad F.A., Aliyan H., Massah A.R.
|
Vol 52, No 1 (2018) |
Design, Synthesis, and Pharmacological Activity of a New Matrix Metalloproteinase-9 Inhibitor |
(Eng)
|
Grigorkevich O.S., Mokrov G.V., Dyabina A.S., Stolyaruk V.N., Tsorin I.B., Ionova E.O., Kryzhanovskii S.A., Gudasheva T.A., Durnev A.D.
|
Vol 51, No 12 (2018) |
Synthesis and Antidepressant Properties of 3-Methyl-7-(1,1-Dioxothietan-3-YL)-8-Cyclohexylamino-1-Ethyl-1H-Purine-2,6(3H,7H)-Dione |
(Eng)
|
Khaliullin F.A., Shabalina Y.V., Davlyatova G.G., Valeeva L.A.
|
Vol 51, No 11 (2018) |
L-Arginine – Cellulose-Acetate-Sulfate Complex and its Influence on Endothelial Dysfunction in Rats |
(Eng)
|
Shakhno E.A., Savitskaya T.A., Grinshpan D.D., Pokrovskaya T.G., Yakushev V.I., Pokrovskii M.V.
|
Vol 51, No 10 (2018) |
Synthesis and Antiradical and Hemorheological Activity of Compounds Based on 2,6-Diisobornyl-4-Methylphenol and Polysaccharides |
(Eng)
|
Plotnikov M.B., Aliev O.I., Sidekhmenova A.V., Popova E.V., Ostrikova O.I., Kuchin A.V., Chukicheva I.Y., Torlopov M.A.
|
Vol 51, No 8 (2017) |
Synthesis, Conversions, and Anti-Monoamine-Oxidase and Anticonvulsant Activity of Ethyl 4′-Amino-5′,8′-Dimethyl-1′H-Spiro[Cyclohexane-1,2′-Naphthalene]-3′-Carboxylate |
(Eng)
|
Grigoryan N.P., Markosyan A.I., Paronikyan R.G., Sukasyan R.S.
|
Vol 51, No 7 (2017) |
Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs |
(Eng)
|
Spasov A.A., Khaliullin F.A., Babkov D.A., Timirkhanova G.A., Kuznetsova V.A., Naumenko L.V., Muleeva D.R., Maika O.Y., Prokhorova T.Y., Sturova E.A.
|
Vol 51, No 6 (2017) |
Protein Glycation During Diabetes Mellitus and the Possibility of its Pharmacological Correction (Review) |
(Eng)
|
Spasov A.A., Solov’eva O.A., Kuznetsova V.A.
|
Vol 51, No 5 (2017) |
Hemocoagulation Activity of Sulfur-Containing Pinane-Type Terpenoids |
(Eng)
|
Kiselev S.V., Nikitina L.E., Startseva V.A., Artemova N.P., Bodrov A.V., Boichuk S.V., Vorontsova M.M., Rakhmatullina A.A., Turaev R.G., Klochkov V.V.
|
Vol 51, No 4 (2017) |
Synthesis, Immunomodulating and Antitumor Activities of Copolymers of Dialkylaminoethyl Methacrylates and Vinylsaccharides |
(Eng)
|
Nazarova O.V., Potapenkova L.S., Stukov A.N., Zolotova Y.I., Zhuravskaya O.N., Nekrasova T.N., Panarin E.F.
|
Vol 51, No 3 (2017) |
The Main Structural Types of Inhibitors of Matrix Metalloproteinases |
(Eng)
|
Kapranov L.E., Reznikov A.N., Klimochkin Y.N.
|
Vol 51, No 2 (2017) |
Web Resources for Discovery and Development of New Medicines |
(Eng)
|
Bezhentsev V.M., Druzhilovskii D.S., Ivanov S.M., Filimonov D.A., Sastry G.N., Poroikov V.V.
|
Vol 51, No 1 (2017) |
2-Thiomorpholino-5-Aryl-6H-1,3,4-Thiadiazine Hydrobromides and Their Ability to Inhibit Nonenzymatic Protein Glycosylation |
(Eng)
|
Sidorova L.P., Tseitler T.A., Emel’yanov V.V., Savateeva E.A., Maksimova N.E., Mochul’skaya N.N., Chereshnev V.A., Chupakhin O.N.
|
Vol 50, No 12 (2017) |
Prediction and Study of Anticonvulsant Properties of Benzimidazole Derivatives |
(Eng)
|
Vasil’ev P.M., Kalitin K.Y., Spasov A.A., Grechko O.Y., Poroikov V.V., Filimonov D.A., Anisimova V.A.
|
Vol 50, No 11 (2017) |
N-Phenylacetylglycyl-L-Proline Ethyl Ester Converts into Cyclo-L-Prolylglycine Showing a Similar Spectrum of Neuropsychotropic Activity |
(Eng)
|
Gudasheva T.A., Kolyasnikova K.N., Kuznetsova E.A., Litvinova S.A., Zolotov N.N., Voronina T.A., Ostrovskaya R.U., Seredenin S.B.
|
Vol 50, No 10 (2017) |
Synthesis and Antibacterial Activity of Hybrid Supramolecular Complexes Based on Tetracycline/Doxycycline and Water-Soluble C60-Fullerene Derivatives |
(Eng)
|
Zhilenkov A.V., Khakina E.A., Troshin P.A., Inchagova K.S., Deryabin D.G.
|
Vol 50, No 9 (2016) |
Synthesis and Analgesic Activity of 9-Aryl-12-Imino-10,11-Dioxatricyclo[5.3.2.01,6]Dodecane-7,8,8-Tricarbonitriles and 3-Aryl-1,1,2,2-Tetracyanocyclopropanes |
(Eng)
|
Mar’yasov M.A., Sheverdov V.P., Nasakin O.E., Makhmudov R.R.
|
Vol 50, No 8 (2016) |
Synthesis of and HIV-1 Integrase Inhibition by 2-[7-(Fluorobenzyloxy)-4-Oxo-4hchromen-3-Yl]-1-Hydroxyimidazoles |
(Eng)
|
Nikitina P.A., Tkach I.I., Knyazhanskaya E.S., Gottikh M.B., Perevalov V.P.
|
Vol 50, No 7 (2016) |
Synthesis, Hydrolysis, and Analgesic Activity of 3-[3-(1-arylethylcarbamoyl)-4-hydroxy-2-oxo-1,2-dihydroquinolin-1-yl]propanenitriles and Their Derivatives |
(Eng)
|
Ukrainets I.V., Taran E.A., Andreeva K.V.
|
Vol 50, No 6 (2016) |
Synthesis and Antidepressant Properties of 2-[3-Methyl-7-(Thietanyl-3)-1-Ethylxanthinyl-8-Thio] Acetic Acid Hydrazides |
(Eng)
|
Valeeva L.A., Davlyatova G.G., Shabalina Y.V., Isakova A.V., Khaliullin F.A., Nikitina I.L.
|
Vol 50, No 4 (2016) |
Synthesis and Anticonvulsive Activity of 5-Pyrrolidin-1-Ylpyrano[4″,3″:4′,5′]Pyrido-3′,2′:4,5]Thieno[3,2-D]Pyrimidine Derivatives |
(Eng)
|
Dashyan S.S., Paronikyan E.G., Noravyan A.S., Paronikyan R.G.
|
Vol 50, No 5 (2016) |
Pharmacological Activity of 4,5-Dihydropyrazole Derivatives (Review) |
(Eng)
|
Korablina D.D., Vorozhtsov N.I., Sviridova L.A., Kalenikova E.I., Medvedev O.S.
|
Vol 50, No 3 (2016) |
Synthesis and Antifungal and Antiviral Activity of N-Benzyl Derivatives of the Tetraene Macrolide Antibiotic Lucensomycin |
(Eng)
|
Belakhov V.V., Garabadzhiu A.V., Kolodyaznaya V.A., Topkova O.V.
|
Vol 50, No 2 (2016) |
Biological Activity of Adamantane-Containing Mono- and Polycyclic Pyrimidine Derivatives* (A Review) |
(Eng)
|
Shokova É.A., Kovalev V.V.
|
Vol 50, No 1 (2016) |
Synthesis and Antibacterial Activity of 3,6-Diaryl-7H-[1,2,4]Triazolo[3,4-b][1,3,4]Thiadiazines |
(Eng)
|
Iradyan M.A., Iradyan N.S., Minasyan N.S., Paronikyan R.V., Stepanyan G.M.
|
Vol 49, No 12 (2016) |
Synthesis, Hydrolytic Stability, and Antileukemic Activity of Azacytidine Nucleoside Analogs |
(Eng)
|
Bozhok T.S., Kalinichenko E.N., Kuz’mitskii B.B., Golubeva M.B.
|
Vol 49, No 11 (2016) |
M-Dinitroaromatic Moiety as a Fragment of Biologically Active Compounds |
(Eng)
|
Piskov V.B., Chernyshev V.P., Karakotov S.D.
|
Vol 49, No 10 (2016) |
Synthesis and Pharmacological Activity of 2,9-Disubstituted Imidazo[1,2-a]Benzimidazole Phenyl- and Alkylthiocarbamides |
(Eng)
|
Anisimova V.A., Zhukovskaya O.N., Spasov A.A., Kuznetsova V.A., Kosolapov V.A., Yakovlev D.S., Solov’eva O.A., Sorotskii D.V., Brigadirova A.A., Vorob’ev E.S.
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