Screening of Some Dioxaboreninopyridine and Aniline Derivatives for Carcinogenic Properties Using a Model Cell-Free System of Regenerating Rat Liver
- 作者: Terent’ev A.1, Syatkin S.2, Kirichuk A.2, Soldatenkov A.2, Kutyakov S.2, Neborak E.2, Shevkun N.2, Kuznetsova O.2, Skorik A.2
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隶属关系:
- N. I. Pirogov Russian National Research Medical University, Ministry of Health of the Russian Federation
- Peoples’ Friendship University of Russia
- 期: 卷 162, 编号 6 (2017)
- 页面: 801-807
- 栏目: Article
- URL: https://journals.rcsi.science/0007-4888/article/view/238585
- DOI: https://doi.org/10.1007/s10517-017-3717-y
- ID: 238585
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详细
We studied the effects of some aniline and dioxaborininopyridine derivatives on the rate of oxidative deamination of putrescine and polyamines in a tissue with high mitotic index. These effects were evaluated quantitatively by measuring diamine oxidase and polyamine oxidase activities in a model cell-free test system of regenerating rat liver tissue. Aniline derivatives exhibited mainly antiproliferative effects and promoted oxidative degradation of putrescine, spermidine, and spermine. Dioxaborininopyridine derivatives inhibited this process, thus exhibiting carcinogenic properties.
作者简介
A. Terent’ev
N. I. Pirogov Russian National Research Medical University, Ministry of Health of the Russian Federation
Email: syata@mail.ru
俄罗斯联邦, Moscow
S. Syatkin
Peoples’ Friendship University of Russia
编辑信件的主要联系方式.
Email: syata@mail.ru
俄罗斯联邦, Moscow
A. Kirichuk
Peoples’ Friendship University of Russia
Email: syata@mail.ru
俄罗斯联邦, Moscow
A. Soldatenkov
Peoples’ Friendship University of Russia
Email: syata@mail.ru
俄罗斯联邦, Moscow
S. Kutyakov
Peoples’ Friendship University of Russia
Email: syata@mail.ru
俄罗斯联邦, Moscow
E. Neborak
Peoples’ Friendship University of Russia
Email: syata@mail.ru
俄罗斯联邦, Moscow
N. Shevkun
Peoples’ Friendship University of Russia
Email: syata@mail.ru
俄罗斯联邦, Moscow
O. Kuznetsova
Peoples’ Friendship University of Russia
Email: syata@mail.ru
俄罗斯联邦, Moscow
A. Skorik
Peoples’ Friendship University of Russia
Email: syata@mail.ru
俄罗斯联邦, Moscow