Antiproliferative activity of ruthenium and osmium clusters with phosphine ligands
- Авторы: Nazarov A.A.1, Nosova Y.N.1, Mikhalev O.V.1, Kovaleva O.N.2, Dyson P.J.3, Milaeva E.R.1
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Учреждения:
- Department of Chemistry, M. V. Lomonosov Moscow State University
- I. M. Sechenov First Moscow State Medical University
- Swiss Federal Institute of Technology in Lausanne
- Выпуск: Том 65, № 2 (2016)
- Страницы: 546-549
- Раздел: Full Articles
- URL: https://journals.rcsi.science/1066-5285/article/view/237279
- DOI: https://doi.org/10.1007/s11172-016-1335-x
- ID: 237279
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Аннотация
New ruthenium and osmium carbonyl clusters with 1,3,5-triaza-7-phosphatricyclo-[3.3.1.13.7]decane and 3,7-diacetyl-1,3,7-triaza-5-phosphabicyclo[3.3.1]nonane ligands were synthesized using Me3NO as an initiator. The data on antiproliferative activity of new compounds against ovarian carcinoma cell cultures A2780 (cisplatin-sensitive) and A2780cisR (cisplatin-resistant) are reported. The dependence of cytotoxicity on the number of phosphine ligands was demonstrated.
Об авторах
A. Nazarov
Department of Chemistry, M. V. Lomonosov Moscow State University
Автор, ответственный за переписку.
Email: nazarov@med.chem.msu.ru
Россия, Build. 3, 1 Leninskie Gory, Moscow, 119991
Yu. Nosova
Department of Chemistry, M. V. Lomonosov Moscow State University
Email: nazarov@med.chem.msu.ru
Россия, Build. 3, 1 Leninskie Gory, Moscow, 119991
O. Mikhalev
Department of Chemistry, M. V. Lomonosov Moscow State University
Email: nazarov@med.chem.msu.ru
Россия, Build. 3, 1 Leninskie Gory, Moscow, 119991
O. Kovaleva
I. M. Sechenov First Moscow State Medical University
Email: nazarov@med.chem.msu.ru
Россия, Build. 2, 8 ul. Trubetskaya, Moscow, 119991
P. Dyson
Swiss Federal Institute of Technology in Lausanne
Email: nazarov@med.chem.msu.ru
Швейцария, Lausanne
E. Milaeva
Department of Chemistry, M. V. Lomonosov Moscow State University
Email: nazarov@med.chem.msu.ru
Россия, Build. 3, 1 Leninskie Gory, Moscow, 119991
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