Synthesis of oxalic acid derivatives and their antitumor activity in experiments in vivo


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A series of amino acid derivatives of oxalic acid were obtained. In combination therapy with conventional cytostatics used in lower doses, the new compounds substantially increase the efficacy of the drugs in the treatment of experimental P388 murine leukemia and some its drug-resistant strains.

作者简介

B. Fedorov

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

S. Goncharova

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

T. Rajevskaya

Institute of Problems of Chemical Physics, Russian Academy of Sciences

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Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

A. Eremeev

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

A. Utenyshev

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

M. Fadeev

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

G. Bogdanov

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

N. Konovalova

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

S. Aldoshin

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: tara@icp.ac.ru
俄罗斯联邦, 1 prosp. Akad. Semenova, Chernogolovka, Moscow Region, Russian Federation, 142432

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