Synthetic approaches to conjugation of aminoadamantanes and carbazoles
- Authors: Sokolov V.B.1, Aksinenko A.Y.1, Epishina T.A.1, Goreva T.V.1, Bachurin S.O.1
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Affiliations:
- Institute of Physiologically Active Substances, Russian Academy of Sciences
- Issue: Vol 66, No 11 (2017)
- Pages: 2110-2114
- Section: Full Article
- URL: https://journals.rcsi.science/1066-5285/article/view/241581
- DOI: https://doi.org/10.1007/s11172-017-1988-0
- ID: 241581
Cite item
Abstract
Five different synthetic approaches for the conjugation of carbazoles with aminoadamantanes via propylene, 2-hydroxypropylene, 1-oxopropylene, 1-oxoethylene and triazole spacers have been proposed. The corresponding mesylate-, acrylate-, chloroacetate-, propargyl-, azido- and epoxy-containing carbazoles and aminoadamantanes were used as the starting compounds.
About the authors
V. B. Sokolov
Institute of Physiologically Active Substances, Russian Academy of Sciences
Author for correspondence.
Email: alaks@ipac.ac.ru
Russian Federation, 1 Severnyi proezd, Chernogolovka, Moscow Region, 142432
A. Yu. Aksinenko
Institute of Physiologically Active Substances, Russian Academy of Sciences
Email: alaks@ipac.ac.ru
Russian Federation, 1 Severnyi proezd, Chernogolovka, Moscow Region, 142432
T. A. Epishina
Institute of Physiologically Active Substances, Russian Academy of Sciences
Email: alaks@ipac.ac.ru
Russian Federation, 1 Severnyi proezd, Chernogolovka, Moscow Region, 142432
T. V. Goreva
Institute of Physiologically Active Substances, Russian Academy of Sciences
Email: alaks@ipac.ac.ru
Russian Federation, 1 Severnyi proezd, Chernogolovka, Moscow Region, 142432
S. O. Bachurin
Institute of Physiologically Active Substances, Russian Academy of Sciences
Email: alaks@ipac.ac.ru
Russian Federation, 1 Severnyi proezd, Chernogolovka, Moscow Region, 142432