Study of Endothelial Protective Activity of Phenol-Derived Thrombin and Arginase-2 Inhibitors KUD-259 and KUD-974
- Authors: Pokrovskii M.V.1, Korokin M.V.1, Kudryavtsev K.V.1, Pokrovskaya T.G.1, Gudyrev O.S.1, Gureev V.V.1, Korokina L.V.1, Povetkin S.V.1
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Affiliations:
- Department of Pharmacology, Medical School, Belgorod State University
- Issue: Vol 163, No 4 (2017)
- Pages: 436-438
- Section: Article
- URL: https://journals.rcsi.science/0007-4888/article/view/238968
- DOI: https://doi.org/10.1007/s10517-017-3822-y
- ID: 238968
Cite item
Abstract
We performed correction of endothelial dysfunction with phenol derivatives KUD-259 and KUD-974 containing heteroatomic and heterocyclic structures. Pharmacological activity of KUD-259 and KUD-974 surpassed that of L-norvaline, a non-selective arginase inhibitor.
About the authors
M. V. Pokrovskii
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Russian Federation, Belgorod
M. V. Korokin
Department of Pharmacology, Medical School, Belgorod State University
Author for correspondence.
Email: mkorokin@mail.ru
Russian Federation, Belgorod
K. V. Kudryavtsev
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Russian Federation, Belgorod
T. G. Pokrovskaya
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Russian Federation, Belgorod
O. S. Gudyrev
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Russian Federation, Belgorod
V. V. Gureev
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Russian Federation, Belgorod
L. V. Korokina
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Russian Federation, Belgorod
S. V. Povetkin
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Russian Federation, Belgorod