Study of Endothelial Protective Activity of Phenol-Derived Thrombin and Arginase-2 Inhibitors KUD-259 and KUD-974
- Autores: Pokrovskii M.1, Korokin M.1, Kudryavtsev K.1, Pokrovskaya T.1, Gudyrev O.1, Gureev V.1, Korokina L.1, Povetkin S.1
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Afiliações:
- Department of Pharmacology, Medical School, Belgorod State University
- Edição: Volume 163, Nº 4 (2017)
- Páginas: 436-438
- Seção: Article
- URL: https://journals.rcsi.science/0007-4888/article/view/238968
- DOI: https://doi.org/10.1007/s10517-017-3822-y
- ID: 238968
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Resumo
We performed correction of endothelial dysfunction with phenol derivatives KUD-259 and KUD-974 containing heteroatomic and heterocyclic structures. Pharmacological activity of KUD-259 and KUD-974 surpassed that of L-norvaline, a non-selective arginase inhibitor.
Sobre autores
M. Pokrovskii
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Rússia, Belgorod
M. Korokin
Department of Pharmacology, Medical School, Belgorod State University
Autor responsável pela correspondência
Email: mkorokin@mail.ru
Rússia, Belgorod
K. Kudryavtsev
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Rússia, Belgorod
T. Pokrovskaya
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Rússia, Belgorod
O. Gudyrev
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Rússia, Belgorod
V. Gureev
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Rússia, Belgorod
L. Korokina
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Rússia, Belgorod
S. Povetkin
Department of Pharmacology, Medical School, Belgorod State University
Email: mkorokin@mail.ru
Rússia, Belgorod