Email this article Synthesis of 1,2-Diazepines by the Bischler–Napieralski Reaction
- Authors: Muratov A.V.1, Grebenyuk S.A.1, Eresko A.B.1
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Affiliations:
- Litvinenko Institute of Physical Organic and Coal Chemistry
- Issue: Vol 54, No 6 (2018)
- Pages: 861-866
- Section: Article
- URL: https://journals.rcsi.science/1070-4280/article/view/218056
- DOI: https://doi.org/10.1134/S1070428018060064
- ID: 218056
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Abstract
A new strategy has been proposed for the synthesis of 5H-[1]benzofuro[2,3-d][1,2]diazepines containing two aryl substituents in the diazepine fragment. The key stage of the synthesis is intramolecular cyclization of the corresponding hydrazides under the Bischler–Napieralski reaction conditions.
About the authors
A. V. Muratov
Litvinenko Institute of Physical Organic and Coal Chemistry
Email: a_eresko77@mail.ru
Ukraine, ul. R. Lyuksemburg 70, Donetsk, 83114
S. A. Grebenyuk
Litvinenko Institute of Physical Organic and Coal Chemistry
Email: a_eresko77@mail.ru
Ukraine, ul. R. Lyuksemburg 70, Donetsk, 83114
A. B. Eresko
Litvinenko Institute of Physical Organic and Coal Chemistry
Author for correspondence.
Email: a_eresko77@mail.ru
Ukraine, ul. R. Lyuksemburg 70, Donetsk, 83114
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