Synthesis, Structure, and Biological Activity of Products of Reactions of 3,4-Dioxohexane-1,6-dioic Acid Esters with 2-Aminophenol
- 作者: Mukovoz P.1, Slepukhin P.2,3, Danilova E.4, Aysuvakova O.1, Glinushkin A.1
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隶属关系:
- All-Russian Research Institute of Phytopathology
- Postovskii Institute of Organic Synthesis, Ural Branch
- Ural Federal University
- Ivanovo State University of Chemistry and Technology
- 期: 卷 88, 编号 7 (2018)
- 页面: 1363-1368
- 栏目: Article
- URL: https://journals.rcsi.science/1070-3632/article/view/222301
- DOI: https://doi.org/10.1134/S1070363218070022
- ID: 222301
如何引用文章
详细
Bioactive derivatives of 1,4-benzoxazine have been prepared via reactions of 3,4-dioxohexane-1,6- dioic (ketipic) acid esters with 2-aminophenol. (2'Z)-2,2'-(2-Hydroxy-2H-1,4-benzoxazin-2-yl-3-ilidene)diacetic acid esters or (2Z)-[2-oxo-2H-1,4-benzoxazin-3(4H)-ylidene]acetic acid esters can be formed depending on the conditions. The structures of the products of dialkyl ketipate esters reactions with 2-aminophenol were determined by means of X-ray diffraction. It has been demonstrated that the prepared compounds exhibit antimycotic activity against test cultures of plant pathogenic fungi (Fusauium sp., Alternarium sp., and Bipolaris soraciniana).
作者简介
P. Mukovoz
All-Russian Research Institute of Phytopathology
编辑信件的主要联系方式.
Email: mpp27@mail.ru
俄罗斯联邦, ul. Institut 5, Bolshie Vyazemy, 143050
P. Slepukhin
Postovskii Institute of Organic Synthesis, Ural Branch; Ural Federal University
Email: mpp27@mail.ru
俄罗斯联邦, Yekaterinburg; Yekaterinburg
E. Danilova
Ivanovo State University of Chemistry and Technology
Email: mpp27@mail.ru
俄罗斯联邦, Ivanovo
O. Aysuvakova
All-Russian Research Institute of Phytopathology
Email: mpp27@mail.ru
俄罗斯联邦, ul. Institut 5, Bolshie Vyazemy, 143050
A. Glinushkin
All-Russian Research Institute of Phytopathology
Email: mpp27@mail.ru
俄罗斯联邦, ul. Institut 5, Bolshie Vyazemy, 143050