Targeted Delivery of Nucleic Acids by Folate-Containing Liposomes into KB-3-1 and HEK 293 Cells


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Targeted cationic liposomes containing folate lipoconjugates with spacer groups of various lengths and natures were prepared; their physicochemical characteristics and their transfection activity towards KB-3-1 and HEK 293 cells were determined. Targeted delivery of plasmid DNA was studied by competitive inhibition of DNA delivery in the presence of free folic acid.

作者简介

E. Shmendel

Lomonosov Institute of Fine Chemical Technologies, MIREA—Russian Technological University

Email: mamaslov@mail.ru
俄罗斯联邦, Moscow, 119571

T. Kabilova

Institute of Chemical Biology and Fundamental Medicine, Siberian Branch, Russian Academy of Sciences

Email: mamaslov@mail.ru
俄罗斯联邦, Novosibirsk, 630090

N. Morozova

Lomonosov Institute of Fine Chemical Technologies, MIREA—Russian Technological University

Email: mamaslov@mail.ru
俄罗斯联邦, Moscow, 119571

M. Zenkova

Institute of Chemical Biology and Fundamental Medicine, Siberian Branch, Russian Academy of Sciences

Email: mamaslov@mail.ru
俄罗斯联邦, Novosibirsk, 630090

M. Maslov

Lomonosov Institute of Fine Chemical Technologies, MIREA—Russian Technological University

编辑信件的主要联系方式.
Email: mamaslov@mail.ru
俄罗斯联邦, Moscow, 119571

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