Synthesis of γ-(Arylamino)butyric Acid Derivatives via Ring-Opening Addition of Arylamines to Cyclopropane-1,1-Dicarboxylates
- 作者: Li S.K.1, Huang L.L.1, Lv Y.D.1, Feng H.D.1
-
隶属关系:
- College of Chemistry and Chemical Engineering
- 期: 卷 55, 编号 9 (2019)
- 页面: 1432-1438
- 栏目: Article
- URL: https://journals.rcsi.science/1070-4280/article/view/221226
- DOI: https://doi.org/10.1134/S1070428019090252
- ID: 221226
如何引用文章
详细
A rapid and efficient catalytic approach has been proposed for the synthesis of dimethyl 2-[2-(aryl-amino)but-3-en-1-yl]- and 2-[2-(arylamino)-2-phenylethyl]malonates in good yields (49-95%) by ring-opening reaction of dimethyl 2-vinyl- and 2-phenylcyclopropane-1,1-dicarboxylates with arylamines in the presence of Yb(III) catalyst under microwave irradiation. The synthesized compounds are convenient precursors to γ-(aryl-amino)butyric acid derivatives.
作者简介
S. Li
College of Chemistry and Chemical Engineering
Email: llhuang999@126.com
中国, Shanghai, 201620
L. Huang
College of Chemistry and Chemical Engineering
编辑信件的主要联系方式.
Email: llhuang999@126.com
中国, Shanghai, 201620
Y. Lv
College of Chemistry and Chemical Engineering
Email: llhuang999@126.com
中国, Shanghai, 201620
H. Feng
College of Chemistry and Chemical Engineering
Email: llhuang999@126.com
中国, Shanghai, 201620
补充文件
