Study of Sedative Tea Phytocomplex within the Framework of Studies Aimed at Creation of a Rectal Dosage Form with Antihistaminic Effect
- Authors: Kulikovskii V.F.1, Zhilyakova E.T.1, Novikov O.O.1, Pisarev D.I.1, Prokushchenko N.V.1, Ivanova L.L.1
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Affiliations:
- Belgorod State National Research University
- Issue: Vol 163, No 6 (2017)
- Pages: 753-756
- Section: Article
- URL: https://journals.rcsi.science/0007-4888/article/view/239234
- DOI: https://doi.org/10.1007/s10517-017-3896-6
- ID: 239234
Cite item
Abstract
We designed a new complex drug with antiallergic effect containing, in addition to the main component loratadine, a phytocomplex for an extra therapeutic effect. A collection of plants with sedative activity is chosen and the optimal agent for extraction of bioactive compounds (40% ethanol) and optimal degree of plant fragmentation are determined. Chemical composition of the sedative tea is evaluated by reverse phase HPLC. The marker components of the species are detected: xanthohumol and isoxanthohumol — Humulus lupulus cone components, Mentha piperita rosmarinic acid, and scutellareine, Menyanthes trifolia element — quercetin-3-rutinoside, and caffeic acid. Standardization of the species by the absolute graduation method in conversion to quercetin-3-rutinoside is suggested.
About the authors
V. F. Kulikovskii
Belgorod State National Research University
Email: pisarev@bsu.edu.ru
Russian Federation, Belgorod
E. T. Zhilyakova
Belgorod State National Research University
Email: pisarev@bsu.edu.ru
Russian Federation, Belgorod
O. O. Novikov
Belgorod State National Research University
Email: pisarev@bsu.edu.ru
Russian Federation, Belgorod
D. I. Pisarev
Belgorod State National Research University
Author for correspondence.
Email: pisarev@bsu.edu.ru
Russian Federation, Belgorod
N. V. Prokushchenko
Belgorod State National Research University
Email: pisarev@bsu.edu.ru
Russian Federation, Belgorod
L. L. Ivanova
Belgorod State National Research University
Email: pisarev@bsu.edu.ru
Russian Federation, Belgorod