N-acyl dopamines induce apoptosis in PC12 cell line via the GPR55 receptor activation


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Resumo

Dopamine amides of arachidonic, docosahexaenoic, and oleic acids were found to induce apoptosis in PC12 cells, which was blocked exclusively by antagonists and preincubation agonists of the receptor GPR55, belonging to the group of non-CB1/CB2 receptors.

Sobre autores

M. Akimov

Shemyakin–Ovchinnikov Institute of Bioorganic Chemistry

Autor responsável pela correspondência
Email: akimovmike@yandex.ru
Rússia, Moscow, 117997

A. Ashba

Shemyakin–Ovchinnikov Institute of Bioorganic Chemistry

Email: akimovmike@yandex.ru
Rússia, Moscow, 117997

N. Gretskaya

Shemyakin–Ovchinnikov Institute of Bioorganic Chemistry

Email: akimovmike@yandex.ru
Rússia, Moscow, 117997

V. Bezuglov

Shemyakin–Ovchinnikov Institute of Bioorganic Chemistry

Email: akimovmike@yandex.ru
Rússia, Moscow, 117997

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