Synthesis of Phosphoisosteres of Amyloid Dipeptide Components

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A simple and effective method was proposed for the synthesis of new phosphinic peptides in free form, structural isosteres of the dipeptide components of beta-amyloid (Aβ42), potential inhibitors of zinc-metalloproteinases.

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作者简介

S. Golovash

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
俄罗斯联邦, Chernogolovka

D. Ivanov

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
俄罗斯联邦, Chernogolovka

A. Borodachev

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
ORCID iD: 0000-0002-3458-5129
俄罗斯联邦, Chernogolovka

V. Shestov

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
俄罗斯联邦, Chernogolovka

M. Dmitriev

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

Email: rvalery@dio.ru
ORCID iD: 0000-0001-8870-195X
俄罗斯联邦, Chernogolovka

V. Ragulin

Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences

编辑信件的主要联系方式.
Email: rvalery@dio.ru
ORCID iD: 0000-0002-3967-1034
俄罗斯联邦, Chernogolovka

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